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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T1878 | XAV-939 | XAV939,NVP-XAV939 | PARP , Wnt/beta-catenin |
XAV-939 (NVP-XAV939) is a Tankyrase (TNKS) inhibitor that inhibits TNKS1 and TNKS2 (IC50=11/4 nM). XAV-939 selectively inhibits Wnt/β-catenin-mediated transcription. |